PerkinElmer

Receptor Ligand Binding

OF

Simplify the development of your assays and the calculation of your results using our radioligands, receptor-transfected cell membranes, and cell lines for radioligand binding applications.

Because radioligands can be directly detected, there is no need to generate intermediate antibodies against your target. Eliminating these antibodies also eliminates the need to optimize an antibody titer and reduces your total assay time by skipping intermediate incubation steps.

You’ll find our receptor-ligand binding reagents and related products perfect matches for all of your receptor binding studies.

 

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"Receptor Ligand Binding" 1-50 of 762 Products and Services

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UNIFILTER-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the Unifilter Harvester.

OMNIFILTER-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the OmniFilter Harvester.

UNIFILTER-96 CELL HARVESTER SS

Speed and simplicity are the primary strengths of the Unifilter Harvester.
LabChip EZ Reader

EZ READER, SHIP LEVEL

The EZ Reader can help to save time and money in your laboratory by identifying the most promising lead candidates faster.

The EZ Reader instrument is available outside the EU. Please contact your local representative for further information.

MICROBETA FILTERMAT-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the FilterMate Harvester. From beginning to end, the FilterMate system is easy to use.

UNIFILTER-24 CELL HARVESTER

Speed and simplicity are the primary strengths of the Unifilter Harvester.

MICROBETA FILTERMAT-24 CELL HARVESTER

Speed and simplicity are the primary strengths of the FilterMate Harvester. From beginning to end, the FilterMate system is easy to use. Need additional information? Click on the tabs in the product details section below.

LH-RH, [125I]-[D-Trp6]-, 10µCi

NEX365 [125I]-[D-Trp6]-LH-RH will be useful for receptor binding studies in cell lines and tissue cultures.
List Price : 1010.00 GBP

Cytisine HCl, [3,5-3H(N)]-, 250µCi (9.25MBq)

Cytisine HCl, [3,5-3H(N)]- will now be made available on a fresh lot schedule. NET1054025UC and NET1054250UC will be available as a fresh lot once a year on March 6 in 2017.
List Price : 1630.00 GBP
PerkinElmer

Membrane Target Systems: Ghrelin (human) membrane preparation, inCHO-K1 cells. 400 Units

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 478.00 GBP

Fractalkine (human, recombinant), 25µCi

NEX368 Fractalkine is the first member of a new class of chemokines. [125I]-Fractalkine binds with high affinity to the CX3CR1 receptor. [125I]-Fractalkine will be useful for the localization and characterization of CXCR1 receptors.
List Price : 2050.00 GBP
PerkinElmer

Membrane Target Systems: GABA B1b in HEK (human) membrane preparation, in HEK-293 cells. 400 Units.

Cell membranes prepared from HEK293 cells stably transfected with human GABA B1b receptor, 400 units.
List Price : 542.00 GBP

Somatostatin, [125I]Tyr11, 10µCi

NEX389 Somatostatin is a cyclic neuropeptide found in the brain, pancreas and hypothalamus and inhibits the release of growth hormone. [125I ] Tyr11 somatostatin binds to the receptors on RINm5F insolinoma cells with high affinity and inhibits the secretion of insulin from pancreatic b cells.
List Price : 874.00 GBP

Cytisine HCl, [3,5-3H(N)]-, 25µCi (925kBq)

Cytisine HCl, [3,5-3H(N)]- will now be made available on a fresh lot schedule. NET1054025UC and NET1054250UC will be available as a fresh lot once a year on March 6 in 2017.
List Price : 454.00 GBP
Receptor-expressing cell lines

ValiScreen Somatostatin sst3 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

Bombesin, [125I]Tyr4-, 10µCi (370kBq)

NEX258 [125I]-Bombesin will be useful as a tracer in RIAs for bombesin like peptides, and as a high specific activity ligand in receptor studies.
List Price : 1010.00 GBP
List Price : 896.00 GBP

Substance P, [125I]Tyr8], 50µCi

Substance P, [125I]Tyr8] is radioiodinated with no carrier added 125I by a lactoperoxidase procedure and is purified by reversed phase HPLC.
List Price : 2390.00 GBP
PerkinElmer

HIS-Tag Beads PS 500 MG

SPA beads for capturing His-tagged proteins and peptides.
List Price : 1110.00 GBP
PerkinElmer

Protein A PS 500 MG Imaging SPA Beads

Protein A-coated SPA beads, for capturing antibodies in proximity-based scintillation assays.
List Price : 295.00 GBP

Lysergic Acid Diethylamide, 2-[125I]iodo-(+), 50µCi

NEX199 Preparations have been shown to be active in binding to the serotonin receptors. LSD affects a large number of the G protein coupled receptors, including all dopamine receptor subtypes, and all adrenoreceptor subtypes, as well as many others. LSD binds to most serotonin receptor subtypes except for 5-HT3 and 5-HT4.
List Price : 2040.00 GBP
Receptor-expressing cell lines

ValiScreen Ghrelin (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

GR 65630, [N-Methyl-3H]-, 25µCi (925kBq)

25 µCi quantities of [N-Methyl-3H]-GR 65630 are available for your research. 
List Price : 428.00 GBP
PerkinElmer

ProfilerPro Kinase Peptide Substrate 5, for LabChip EZ Reader

Fluorescently-labelled peptide substrate 5 for kinase assays (inhibiton, target discovery, lead optimization)
List Price : 555.00 GBP
Receptor-expressing cell lines

Neuropeptide FF NPFF1 ValiScreen Cell Line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

Membrane Target Systems: Dopamine D42 (human) membrane preparation

Cell membranes prepared from cells stably-transfected with Dopamine D42 (human) receptor, in CHO-K1 cells.
List Price : 568.00 GBP

MESULERGINE, [N-METHYL-3H]-, 250 µCi

250 µCi quantities of tritiated Mesulergine are available for your research.
List Price : 1350.00 GBP
List Price : 771.00 GBP
PerkinElmer

Anti-sheep YSI 500 MG

Anti-sheep-coated SPA beads, for capturing sheep IgG antibodies in proximity-based radiometric scintillation assays.
List Price : 478.00 GBP

4-DAMP, [N-Methyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [N-Methyl-3H]-4-DAMP are available for your research.
List Price : 1590.00 GBP

Prazosin, [7-Methoxy-3H]-, 25µCi (925kBq)

25 µCi quantities of [7-Methoxy-3H]-Prazosin are available for your research.
List Price : 532.00 GBP
Receptor-expressing cell lines

ValiScreen Histamine H2 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

WGA PS Imaging Beads 50 MG

WGA-coated SPA beads, for capturing cell membranes in proximity-based scintillation assays.
List Price : 28.00 GBP
PerkinElmer

Membrane Target Systems: Thromboxane TP (human) membrane preparation

Cell membranes prepared from cells stably-transfected with human Thromboxane TP receptor, in HEK-293 cells.
List Price : 542.00 GBP

Nicotine, L-(-)-[N-Methyl-3H]-, 25µCi (925kBq)

25 µCi quantities of L-(-)-[N-Methyl-3H]-Nicotine are available for your research.
List Price : 373.00 GBP
PerkinElmer

Membrane Target Systems: Adenosine A1 (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 542.00 GBP
PerkinElmer

PDE Substrate iFL-cGMP, for LabChip EZ Reader

Fluorescently-labelled cGMP for Phosphodiesterase Assays (Enyzme inhibiton, target discovery, lead optimization)
List Price : 555.00 GBP

U-69,593, [Phenyl-3,4-3H]-, 25µCi (925kBq)

25 µCi quantities of [Phenyl-3, 4-3H]-U-69,593 are available for your research.
List Price : 527.00 GBP
PerkinElmer

Protein A PVT Beads 25X500MG

Protein A-coated SPA beads, for capturing antibodies in proximity-based radiometric scintillation assays.
List Price : 11880.00 GBP

Peptide YY, (Porcine), ([125I]-PYY), 50µCi

NEX240 Synthetic Peptide YY is radioiodinated with no-carrier-added 125I using a modification of the chloramine-T method.
List Price : 2250.00 GBP
PerkinElmer

Membrane Target Systems: Neuromedin U NMU1 (FM3) (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 542.00 GBP
PerkinElmer

Membrane Target Systems: Muscarinic M4 (human) membrane preparation

Cell membranes prepared from cells stably-transfected with human Muscarinic M4 receptor, in CHO-K1 cells.
List Price : 542.00 GBP

MDL105,519, [3H]

250 µCi quantities of [3H]-MDL105,519 are available for your research.
List Price : 2000.00 GBP
Receptor-expressing cell lines

ValiScreen Nicotinic HM74a (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
Receptor-expressing cell lines

ValiScreen Chemokine CXCR2 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

Membrane Target Systems: Serotonin 5HT-2A (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 542.00 GBP

"Receptor Ligand Binding" 1-50 of 762 Products and Services

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