PerkinElmer

Receptor Ligand Binding

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Simplify the development of your assays and the calculation of your results using our radioligands, receptor-transfected cell membranes, and cell lines for radioligand binding applications.

Because radioligands can be directly detected, there is no need to generate intermediate antibodies against your target. Eliminating these antibodies also eliminates the need to optimize an antibody titer and reduces your total assay time by skipping intermediate incubation steps.

You’ll find our receptor-ligand binding reagents and related products perfect matches for all of your receptor binding studies.

 

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"Receptor Ligand Binding" 1-50 of 764 Products and Services

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MICROBETA FILTERMAT-24 CELL HARVESTER

Speed and simplicity are the primary strengths of the FilterMate Harvester. From beginning to end, the FilterMate system is easy to use. Need additional information? Click on the tabs in the product details section below.

UNIFILTER-96 CELL HARVESTER SS

Speed and simplicity are the primary strengths of the Unifilter Harvester.

MICROBETA FILTERMAT-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the FilterMate Harvester. From beginning to end, the FilterMate system is easy to use.

UNIFILTER-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the Unifilter Harvester.

UNIFILTER-24 CELL HARVESTER

Speed and simplicity are the primary strengths of the Unifilter Harvester.
LabChip EZ Reader

EZ READER, SHIP LEVEL

The EZ Reader can help to save time and money in your laboratory by identifying the most promising lead candidates faster.

OMNIFILTER-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the OmniFilter Harvester.

(+)-Pentazocine, [Ring-1,3-3H]-,250µCi (9.25MBq)

250 µCi quantities of [Ring-1, 3-3H]-(+)-Pentazocine are available for your research.
List Price : 1540.00 GBP

Prazosin, [7-Methoxy-3H]-, 25µCi (925kBq)

25 µCi quantities of [7-Methoxy-3H]-Prazosin are available for your research.
List Price : 532.00 GBP

DICLOFENAC SODIUM[PHENYLACETIC ACID RING- U-14C]

50 µCi quantities of [Phenylacetic Acid Ring - 14C(U)]-Diclofenac Sodium are available for your research.
List Price : 1560.00 GBP
List Price : 1050.00 GBP

Propranolol, L-[4-3H]-, 250µCi (9.25MBq)

250 µCi quantities of tritiated L-propranolol are available for your research.
List Price : 1000.00 GBP
PerkinElmer

Membrane Target Systems: Opioid Delta (human) membrane preparation

Cell membranes prepared from cells stably-transfected with human Opioid Delta receptor, in CHO-K1 cells.
List Price : 542.00 GBP
PerkinElmer

Membrane Target Systems: Serotonin 5HT-2A (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 542.00 GBP

Lysergic Acid Diethylamide, 2-[125I]iodo-(+), 10µCi

NEX199 Preparations have been shown to be active in binding to the serotonin receptors. LSD affects a large number of the G protein coupled receptors, including all dopamine receptor subtypes, and all adrenoreceptor subtypes, as well as many others. LSD binds to most serotonin receptor subtypes except for 5-HT3 and 5-HT4.
List Price : 851.00 GBP
Receptor-expressing cell lines

ValiScreen Leukotriene BLT1 (LTB4R1) (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

Nisoxetine Hydrochloride, [N-Methyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [N-Methyl-3H]-Nisoxetine Hydrochloride are available for your research.
List Price : 1640.00 GBP
PerkinElmer

ProfilerPro Kinase Peptide Substrate 1, for LabChip EZ Reader

Fluorescently-labelled peptide substrate 1 for kinase assays (inhibiton, target discovery, lead optimization)
List Price : 555.00 GBP

Acetylcholine Iodide, [acetyl-3H], 1mCi (37MBq)

1 mCi quantities of Acetylcholine Iodide, [acetyl-3H]- are available for your research.
List Price : 568.00 GBP
PerkinElmer

Membrane Target Systems: Cannabinoid CB1 (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 542.00 GBP
PerkinElmer

Membrane Target Systems: Serotonin 5HT-2C (e) (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 542.00 GBP

Endothelin-1 (human, porcine), [125I]Tyr13, 5µCi

NEX259 [125I]-ET-1 will be useful as a tracer in RIA's for endothelin, and as a high specific activity ligand in receptor studies encompassing the areas of vasoconstriction and stroke, smooth muscle and renal function, and in the study of neurotransmitters in the CNS.
List Price : 882.00 GBP
Receptor-expressing cell lines

ValiScreen Serotonin 5HT-1A (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

ProfilerPro Kinase Selectivity Assay Plate Kit 8, for LabChip EZ Reader

Kit consist of matched pairs of 384-well kinase-assay and substrate plates. Each assay plate contains 24 different predispensed frozen kinases. Substrate plates contain the appropriate fluorescent labeled peptides and ATP.
List Price : 1190.00 GBP

Lysergic Acid Diethylamide, 2-[125I]iodo-(+), 250µCi

NEX199 Preparations have been shown to be active in binding to the serotonin receptors. LSD affects a large number of the G protein coupled receptors, including all dopamine receptor subtypes, and all adrenoreceptor subtypes, as well as many others. LSD binds to most serotonin receptor subtypes except for 5-HT3 and 5-HT4.
List Price : 4640.00 GBP

PK 11195, [N-Methyl-3H]-, 25µCi (925kBq)

25 µCi quantities of [N-Methyl-3H]-PK 11195 are available for your research.
List Price : 462.00 GBP

Batrachotoxinin A 20-α-Benzoate, [Benzoyl-2,5-3H]-, 250µCi (9.25MBq)

Batrachotoxinin A 20-α-Benzoate, [Benzoyl-2,5-3H]- will now be made available on a fresh lot schedule. NET876100UC and NET876250UC will be available as a fresh lot once a year on March 15 in 2017.
PerkinElmer

Membrane Target Systems: Neurotensin NTS1(Leu194) (human) membrane preparation, in CHO-K1 cells. 400 Units.

Cell membranes prepared from CHO-K1 cells stably-transfected with human neurotensin NTS1 (Leu194) receptor, 400 units.
List Price : 527.00 GBP
Receptor-expressing cell lines

ValiScreen Adrenergic beta 2 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

Membrane Target Systems: Somatostatin sst4 (human) membrane preparation

Cell membranes prepared from cells stably-transfected with human Somatostatin sst4 receptor, in HEK-293 cells.
List Price : 542.00 GBP

DELFIA Eu-N1 ITC chelate & Eu standard, 1 mg

DELFIA® Europium labeling chelate and Europium standard for labeling your own biomolecules for use in DELFIA time-resolved fluorescence assays. The ITC chelate reacts with free amine groups in the target biomolecule.
List Price : 1280.00 GBP
Receptor-expressing cell lines

ValiScreen Purinergic P2Y6 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

Ro 15-1788, [N-Methyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [N-Methyl-3H]-Ro 15-1788 are available for your research.
List Price : 1640.00 GBP
PerkinElmer

Membrane Target Systems: Serotonin 5HT-6 (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 542.00 GBP

Endothelin-1 (human, porcine), [125I]Tyr13, 10µCi

NEX259 [125I]-ET-1 will be useful as a tracer in RIA's for endothelin, and as a high specific activity ligand in receptor studies encompassing the areas of vasoconstriction and stroke, smooth muscle and renal function, and in the study of neurotransmitters in the CNS.
List Price : 1220.00 GBP

SCH 23390, [N-Methyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [N-Methyl-3H]-SCH 23390 are available for your research.
List Price : 1320.00 GBP

Bombesin (6-14), D-Tyr6[125I], 10µCi

NEX377 [D-Tyr6[125I]-, βAla11, Phe13, Nle14]-Bombesin (6-14) is a high affinity agonist to the human Orphan Bombesin Receptor Subtype 3 (hBRS-3).
[D-Tyr6[125I]-, bAla11, Phe13, Nle14]-Bombesin (6-14) will be a useful tool to study the pharmacology of this orphan receptor as well as the natural ligand for this receptor.
List Price : 1230.00 GBP
PerkinElmer

WGA PEI TYPE B PVT 2G

WGA-coated SPA beads, for capturing cell membranes in proximity-based radiometric scintillation assays.
List Price : 1910.00 GBP
PerkinElmer

Membrane Target Systems: Serotonin 5-HT1a (human) membrane preparation

Cell membranes prepared from cells stably-transfected with human Serotonin 5-HT1a receptor, in HEK-293 cells.
List Price : 542.00 GBP

Enkephalin, [Tyrosyl-2,6-3H(N)]- (2-D-Penicillamine, 5-D-Penicillamine) (DPDPE), 50µCi (1.85MBq)

50 µCi quantities of [Tyrosyl-2, 6-3H(N)]-Enkephalin (2-D-Penicillamine, 5-D-Penicillamine), (DPDPE) are available for your research.
List Price : 621.00 GBP

RTI-55, [125I]-, 25µCi (925kBq)

NEX272 [125I]-RTI-55 is an excellent radioligand for the study of the dopamine transporter sites using either tissue homogenates or autoradiographic methods--especially in regions of low receptor density.
List Price : 874.00 GBP

Sphingosine-1-phosphate, 33P

Sphingosine-1-phosphate is a bioactive lipid and can be used as an endogenous ligand in sphingosine-1-phosphate (S1P) receptor binding assays.
Price Range : 11480.00 GBP - 28400.00 GBP
PerkinElmer

ProfilerPro Kinase Selectivity Assay Plate Kit 9, for LabChip EZ Reader

Kit consist of matched pairs of 384-well kinase-assay and substrate plates. Each assay plate contains 24 different predispensed frozen kinases. Substrate plates contain the appropriate fluorescent labeled peptides and ATP.
List Price : 985.00 GBP

Goat anti-rabbit IgG, [125I], 100µCi (3.7MBq)

Affinity purified goat anti-rabbit IgG is radioiodinated with no carrier added 125I using a modification of the Hunter and Greenwood method1 and is purified by gel filtration chromatography. This method predominantly labels tyrosine residues.
List Price : 774.00 GBP
List Price : 2600.00 GBP
Receptor-expressing cell lines

ValiScreen Serotonin 5HT-5A (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

α-Dendrotoxin [125I] 5 µCi

NEX434 [125I]- α-Dendrotoxinsare a class of neurotoxins produced by mamba snakes that block particular subtypes of voltage-gated potassium channels in neurons. Dendrotoxins enhance the release of acetylcholine at neuromuscular junctions.
List Price : 1020.00 GBP

Nicotine, L-(-)-[N-Methyl-3H]-, 1mCi (37MBq)

1 mCi quantities of L-(-)-[N-Methyl-3H]-Nicotine are available for your research.
List Price : 2880.00 GBP

Cocaine, Levo-[benzoyl-3,4-3H(N)]-

100 µCi and 250 µCi quantities of Levo-[benzoyl-3, 4-3H(N)]-Cocaine are available for your research. 
List Price : 2010.00 GBP
List Price : 972.00 GBP

"Receptor Ligand Binding" 1-50 of 764 Products and Services

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