PerkinElmer

Receptor Ligand Binding

OF

Simplify the development of your assays and the calculation of your results using our radioligands, receptor-transfected cell membranes, and cell lines for radioligand binding applications.

Because radioligands can be directly detected, there is no need to generate intermediate antibodies against your target. Eliminating these antibodies also eliminates the need to optimize an antibody titer and reduces your total assay time by skipping intermediate incubation steps.

You’ll find our receptor-ligand binding reagents and related products perfect matches for all of your receptor binding studies.

 

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"Receptor Ligand Binding" 1-50 of 780 Products and Services

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OMNIFILTER-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the OmniFilter Harvester.

UNIFILTER-96 CELL HARVESTER SS

Speed and simplicity are the primary strengths of the Unifilter Harvester.

MICROBETA FILTERMAT-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the FilterMate Harvester. From beginning to end, the FilterMate system is easy to use.
LabChip EZ Reader

EZ READER, SHIP LEVEL

The EZ Reader can help to save time and money in your laboratory by identifying the most promising lead candidates faster.

UNIFILTER-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the Unifilter Harvester.

MICROBETA FILTERMAT-24 CELL HARVESTER

Speed and simplicity are the primary strengths of the FilterMate Harvester. From beginning to end, the FilterMate system is easy to use. Need additional information? Click on the tabs in the product details section below.

UNIFILTER-24 CELL HARVESTER

Speed and simplicity are the primary strengths of the Unifilter Harvester.
List Price : 1050.00 GBP

AH5183, L-[PIPERIDINYL-3,4-3H]-(VESAMICOL), 250 µCi

Vesamicol (AH5183) an acetylcholine uptake blocker in presynaptic vesicles,reduces the apparent activity of cholinergic neurons, but does not act at the post-synaptic ACh receptor. Vesamicol is a unique tool for investigating presynaptic mechanisms in cholinergic nerve terminals.
List Price : 591.00 GBP
List Price : 1710.00 GBP

AF-DX 384, [2,3-Dipropylamino-3H]-, 250µCi (9.25MBq)

250 µCi quantities of AF-DX 384, [2, 3-Dipropylamino-3H]- are available for your research.
List Price : 1480.00 GBP

8-Hydroxy-DPAT, [Propyl-2,3-ring-1,2,3-3H]-, 1mCi (37MBq)

1 mCi quantities of [Propyl-2, 3-ring-1, 2, 3-3H]-8-Hydroxy-DPAT are available for your research.
List Price : 2210.00 GBP

Lysergic Acid Diethylamide, 2-[125I]iodo-(+), 10µCi

NEX199 Preparations have been shown to be active in binding to the serotonin receptors. LSD affects a large number of the G protein coupled receptors, including all dopamine receptor subtypes, and all adrenoreceptor subtypes, as well as many others. LSD binds to most serotonin receptor subtypes except for 5-HT3 and 5-HT4.
List Price : 851.00 GBP

PN200-110, (+)-[5-Methyl-3H]-, 250µCi (9.25MBq)

Note: This product will be discontinued from our catalog portfolio on January 1, 2017.
List Price : 1450.00 GBP

Quinpirole, [N-Propyl-3H]-, 25µCi (925kBq)

Note: This product will be discontinued from our catalog portfolio on January 1, 2017.
List Price : 444.00 GBP

Lysergic Acid Diethylamide, 2-[125I]iodo-(+), 50µCi

NEX199 Preparations have been shown to be active in binding to the serotonin receptors. LSD affects a large number of the G protein coupled receptors, including all dopamine receptor subtypes, and all adrenoreceptor subtypes, as well as many others. LSD binds to most serotonin receptor subtypes except for 5-HT3 and 5-HT4.
List Price : 2040.00 GBP
List Price : 1760.00 GBP

Batrachotoxinin A 20-α-Benzoate, [Benzoyl-2,5-3H]-, 100µCi (3.7MBq)

Batrachotoxinin A 20-α-Benzoate, [Benzoyl-2,5-3H]- will now be made available on a fresh lot schedule. NET876100UC and NET876250UC will be available as a fresh lot once a year on March 15 in 2017.
Receptor-expressing cell lines

ValiScreen Histamine H1 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

Verapamil Hydrochloride, [N-Methyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [N-Methyl-3H]-Verapamil Hydrochloride are available for your research.
List Price : 1580.00 GBP

Lysergic Acid Diethylamide, 2-[125I]iodo-(+), 250µCi

NEX199 Preparations have been shown to be active in binding to the serotonin receptors. LSD affects a large number of the G protein coupled receptors, including all dopamine receptor subtypes, and all adrenoreceptor subtypes, as well as many others. LSD binds to most serotonin receptor subtypes except for 5-HT3 and 5-HT4.
List Price : 4640.00 GBP
Receptor-expressing cell lines

ValiScreen Prostanoid EP2 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

Retinoic Acid, [11,12-3H]9-cis-

cis-Retinoic Acid may be used in dermatological applications.
List Price : 1600.00 GBP

UniFilter-96 GF/C PEI Coated Plates

PEI-coated GF/C glassfibre filter-bottom 96-well microplate, for receptor binding and cell harvesting assays using a vacuum manifold.
List Price : 572.00 GBP

CGP 39653, [Propyl-2,3,3H]-, 25µCi (925kBq)

25 µCi quantities of [Propyl-2, 3, 3H]-CGP 39653 are available for your research
List Price : 444.00 GBP
PerkinElmer

Membrane Target Systems: Histamine H1 (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 542.00 GBP

8-Hydroxy-DPAT, [Propyl-2,3-ring-1,2,3-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [Propyl-2, 3-ring-1, 2, 3-3H]-8-Hydroxy-DPAT are available for your research.
List Price : 914.00 GBP
Receptor-expressing cell lines

ValiScreen Neurokinin NK2 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

GBR 12935, [Propylene-2,3-3H]-, 1mCi (37MBq)

1 mCi quantities of tritiated GBR 12935 are available for your research.
List Price : 4600.00 GBP

TCP, [Piperdyl-3,4-3H(N)]-

25 µCi quantities of [Piperidyl-3,4-3H(N)]-TCP are available for your research.
List Price : 432.00 GBP

(+)-Pentazocine, [Ring-1,3-3H]-, 25µCi (925kBq)

25 µCi quantities of [Ring-1, 3-3H]-(+)-Pentazocine are available for your research.
List Price : 473.00 GBP
Receptor-expressing cell lines

ValiScreen Cannabinoid CB1 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

Rosiglitazone, DL- [3H]-

100 µCi quantities of tritiated DL-Rosiglitazone are available for your research.
List Price : 865.00 GBP
PerkinElmer

Membrane Target Systems: Angiotensin AT2 (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 542.00 GBP

UniFilter-96 GF/B PEI Coated Plates - Case of 50

PEI-coated GF/B glassfibre filter-bottom 96-well microplate, for receptor binding and cell harvesting assays using a vacuum manifold.
List Price : 572.00 GBP
List Price : 1760.00 GBP

Clonidine Hydrochloride, [Benzene Ring-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [Benzene Ring-3H]-Clonidine Hydrochloride are available for your research.
List Price : 871.00 GBP
PerkinElmer

Membrane Target Systems: Serotonin 5HT-2C (e) (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 542.00 GBP
List Price : 1580.00 GBP
PerkinElmer

Membrane Target Systems: Endothelin ETB (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 542.00 GBP

Ghrelin (human), [His[125I]], 25µCi

NEX388 Ghrelin is an acylated endogenous peptide which stimulates the release of growth hormone from the pituitary through an orphan G-protein-coupled receptor (GHS-R)7. Ghrelin is an appetite inducing hormone produced in the stomach and the upper portion of the small intestine. [ [125I]His ]Ghrelin (human), binds to GHS-R with high affinity.
List Price : 2540.00 GBP

Quinpirole, [N-Propyl-3H]-, 250µCi (9.25MBq)

Note: This product will be discontinued from our catalog portfolio on January 1, 2017.
List Price : 1600.00 GBP
Receptor-expressing cell lines

ValiScreen Somatostatin sst4 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

Nitrendipine, [5-Methyl-3H]-, 25µCi (925kBq)

25 µCi quantities of tritiated Nitrendipine are available for your research.
List Price : 550.00 GBP

Dihydroxyphenylethylamine, 3,4-[7-3H]-, 250µCi (9.25MBq)

250 µCi quantities of 3, 4-[7-3H]-Dihydroxyphenylethylamine (Dopamine) are available for your research.
List Price : 493.00 GBP
PerkinElmer

WGA PEI TYPE A PVT 25 X 2G

WGA-coated SPA beads, for capturing cell membranes in proximity-based radiometric scintillation assays.
List Price : 31850.00 GBP

α-Bungarotoxin, [125I]-Tyr54-, 50µCi (1.85MBq)

α-bungarotoxin extracted from venom of the Taiwanese banded krait (Bungarus multicinctus) binds the nicotinic acetylcholine receptor found at the neuromuscular junction and the 7 nicotinic acetylcholine receptor in the brain.
List Price : 548.00 GBP
List Price : 3850.00 GBP

"Receptor Ligand Binding" 1-50 of 780 Products and Services

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