PerkinElmer

Receptor Ligand Binding

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Simplify the development of your assays and the calculation of your results using our radioligands, receptor-transfected cell membranes, and cell lines for radioligand binding applications.

Because radioligands can be directly detected, there is no need to generate intermediate antibodies against your target. Eliminating these antibodies also eliminates the need to optimize an antibody titer and reduces your total assay time by skipping intermediate incubation steps.

You’ll find our receptor-ligand binding reagents and related products perfect matches for all of your receptor binding studies.

 

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"Receptor Ligand Binding" 1-50 of 764 Products and Services

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MICROBETA FILTERMAT-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the FilterMate Harvester. From beginning to end, the FilterMate system is easy to use.

UNIFILTER-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the Unifilter Harvester.

MICROBETA FILTERMAT-24 CELL HARVESTER

Speed and simplicity are the primary strengths of the FilterMate Harvester. From beginning to end, the FilterMate system is easy to use. Need additional information? Click on the tabs in the product details section below.

OMNIFILTER-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the OmniFilter Harvester.

UNIFILTER-96 CELL HARVESTER SS

Speed and simplicity are the primary strengths of the Unifilter Harvester.
LabChip EZ Reader

EZ READER, SHIP LEVEL

The EZ Reader can help to save time and money in your laboratory by identifying the most promising lead candidates faster.

The EZ Reader instrument is no longer available in EU. Please contact your local representative for further information.

UNIFILTER-24 CELL HARVESTER

Speed and simplicity are the primary strengths of the Unifilter Harvester.

(+/-)Epibatidine, [5,6-Bicycloheptyl-3H]-, 25µCi (925kBq)

25 µCi quantities of [+/-] [5, 6-Bicycloheptyl-3H]-Epibatidine are available for your research.
List Price : 1310.00 GBP

Dihydroxyphenylethylamine [2,5,6,7,8-3H] (Dopamine)

Dopamine receptors have key roles in many processes, including the control of motivation, learning, and fine motor movement, as well as modulation of neuroendocrine signaling.
List Price : 1310.00 GBP
PerkinElmer

Membrane Target Systems: Cannabinoid CB2 (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 542.00 GBP
List Price : 1220.00 GBP
PerkinElmer

Membrane Target Systems: Cannabinoid CB1 (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 542.00 GBP
List Price : 2600.00 GBP

(-)-CGP-12177, [5,7-3H]-, 250µCi (9.25MBq)

250 µCi quantities of (-)-CGP-12177, [5,7-3H]- are available for your research.
List Price : 953.00 GBP

(-)-CGP-12177, [5,7-3H]-, 25µCi (925kBq)

25 µCi quantities of (-)-CGP-12177, [5,7-3H]- are available for your research.
List Price : 390.00 GBP

INSULIN (porcine), [125I], 10µCi (370kBq), Specific Activity:80-120µCi (2.96-4.44MBq)/µg

NEX104 Insulin (porcine) is radioiodinated with no carrier added 125I using a modification of the Hunter and Greenwood method and purified by ion-exchange column chromatography. This method predominantly labels tyrosine residues.
List Price : 806.00 GBP
List Price : 1050.00 GBP

(+)-Pentazocine, [Ring-1,3-3H]-, 1mCi (37MBq)

1 mCi quantities of [Ring-1, 3-3H]-(+)-Pentazocine are available for your research.
List Price : 3690.00 GBP

Sphingosine-1-phosphate, 33P

Sphingosine-1-phosphate is a bioactive lipid and can be used as an endogenous ligand in sphingosine-1-phosphate (S1P) receptor binding assays.
Price Range : 11480.00 GBP - 28400.00 GBP
Receptor-expressing cell lines

ValiScreen Cannabinoid CB2 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

Membrane Target Systems: Endothelin ETB (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 542.00 GBP

Ketanserin Hydrochloride (R41 468), [Ethylene-3H]-, 25µCi (925kBq)

25 µCi quantities of tritiated Ketanserin hydrochloride are available for your research.
List Price : 468.00 GBP

Peptide YY, (Porcine), ([125I]-PYY), 10µCi

NEX240 Synthetic Peptide YY is radioiodinated with no-carrier-added 125I using a modification of the chloramine-T method.
List Price : 974.00 GBP

Apamin [125I]His18-NH2, 50µCi

NEX242 [125I]-Apamin is a K+ channel antagonist and can be used in the detection and quantification of K+ channel receptors. [125I]-Apamin has been used in receptor binding assays and in autoradiography.
List Price : 1440.00 GBP
List Price : 2290.00 GBP
List Price : 977.00 GBP

BRL-43694, [9-Methyl-3H]-, 250µCi (9.25MBq)

Please note that as of Jan 1, 2016, this product will be discontinued.
List Price : 1730.00 GBP
PerkinElmer

Membrane Target Systems: Nicotinic membrane preparation

Cell membranes prepared from IMR32 cells containing human endogenous Nicotinic receptor.
List Price : 542.00 GBP

AB-MECA, [125I]-(4-Amino-3-[125I]iodobenzyl-5`-N-)-, 50µCi

AB-MECA is radioiodinated with no carrier added 125I using a modification of the Hunter and Greenwood method and is purified by reversed phase HPLC.
List Price : 2240.00 GBP
PerkinElmer

Membrane Target Systems: Bombesin BB1 (human) membrane preparation

Cell membranes prepared from cells stably-transfected with Bombesin BB1 (human) receptor, in CHO-K1 cells.
List Price : 542.00 GBP

DOFETILIDE, [N-METHYL-3H], 100 µCi

100 µCi quantities of tritiated Dofetilide are available for your research.
List Price : 1200.00 GBP
PerkinElmer

Membrane Target Systems: K562 cells membranes

Wild Type Subtype K562 Control Membrane frozen suspension cell membrane. Shipped on dry ice.
List Price : 323.00 GBP

Endothelin-1 (human, porcine), [125I]Tyr13, 50µCi

NEX259 [125I]-ET-1 will be useful as a tracer in RIA's for endothelin, and as a high specific activity ligand in receptor studies encompassing the areas of vasoconstriction and stroke, smooth muscle and renal function, and in the study of neurotransmitters in the CNS.
List Price : 2430.00 GBP
PerkinElmer

Membrane Target Systems: Cannabinoid CB2 (human) membrane preparation

Cell membranes prepared from cells stably-transfected with human Cannabinoid CB2 receptor, in HEK-293 cells.
List Price : 542.00 GBP

Lysergic Acid Diethylamide, 2-[125I]iodo-(+), 50µCi

NEX199 Preparations have been shown to be active in binding to the serotonin receptors. LSD affects a large number of the G protein coupled receptors, including all dopamine receptor subtypes, and all adrenoreceptor subtypes, as well as many others. LSD binds to most serotonin receptor subtypes except for 5-HT3 and 5-HT4.
List Price : 2040.00 GBP

(+/-)Epibatidine, [5,6-Bicycloheptyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [+/-] [5, 6-Bicycloheptyl-3H]-Epibatidine are available for your research. 
List Price : 3080.00 GBP
PerkinElmer

Protein A PS 500 MG Imaging SPA Beads

Protein A-coated SPA beads, for capturing antibodies in proximity-based scintillation assays.
List Price : 295.00 GBP

Insulin (human, recombinant), [125I], 10 µCi

[125I]-Insulin (h) is suitable for the use in radioimmunoassay as well as receptor binding assay. [125I]-Insulin (h) is radioiodinated with no carrier added 125I using the LPO iodination procedure and is purified by reversed phase HPLC.
List Price : 1050.00 GBP
PerkinElmer

Streptavidin PVT 50MG

Streptavidin-coated SPA beads, for capturing biotinylated biomolecules in proximity-based radiometric scintillation assays.
List Price : 160.00 GBP

Lysergic Acid Diethylamide, 2-[125I]iodo-(+), 10µCi

NEX199 Preparations have been shown to be active in binding to the serotonin receptors. LSD affects a large number of the G protein coupled receptors, including all dopamine receptor subtypes, and all adrenoreceptor subtypes, as well as many others. LSD binds to most serotonin receptor subtypes except for 5-HT3 and 5-HT4.
List Price : 851.00 GBP

Calcitonin [Tyr22] (salmon), [125I] 10 µCi

NEX423 [125I]-Calcitonin, [Tyr22] (s) is suitable for the use in radioimmunoassay as well as in the radio-receptor assay.
List Price : 859.00 GBP

Butyl Bicyclophosphorothionate, Tertiary-[35S]-, 100µCi (3.7MBq), Ethanol under nitrogen

35S t-butyl bicyclophosphorothionate (TBPS) is a picrotoxinin analog cage-convulsant that binds GABAA receptors with high affinity and high specificity. Its binding site is closely associated with the chloride ion channel, leading to its classification as a chloride ion channel blocking ligand.
List Price : 1530.00 GBP
PerkinElmer

Membrane Target Systems: Opioid Delta (human) membrane preparation

Cell membranes prepared from cells stably-transfected with human Opioid Delta receptor, in CHO-K1 cells.
List Price : 542.00 GBP

QUISQUALIC ACID, [3H]

50 µCi quantities of [3H]-Quisqualic Acid are available for your research. This product has a scheduled release date for the third Monday in September.
List Price : 1290.00 GBP
PerkinElmer

Polylysine PS Imaging Bead 500 MG

Poly-L-lysine SPA beads enhance the binding of negatively-charged membranes to beads.
List Price : 238.00 GBP
PerkinElmer

Membrane Target Systems: Histamine H2 (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 542.00 GBP
List Price : 1890.00 GBP
PerkinElmer

Membrane Target Systems: Neurotensin NTS1 (human) membrane preparation

Cell membranes prepared from cells stably-transfected with human Neurotensin NTS1 receptor, in HEK-293 cells.
List Price : 542.00 GBP
PerkinElmer

Membrane Target Systems: Somatostatin sst4 (human) membrane preparation

Cell membranes prepared from cells stably-transfected with human Somatostatin sst4 receptor, in HEK-293 cells.
List Price : 542.00 GBP
Receptor-expressing cell lines

ValiScreen KiSS-1 (GPR54) (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

"Receptor Ligand Binding" 1-50 of 764 Products and Services

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